Found 64 of ic50 for ACETYLCHOLINE RECEPTOR SUBUNIT EPSILON
having polymerids = 50000820,50000821 and
complexids = 50000437,50000466,50005823,50014578
having polymerids = 50000820,50000821 and
complexids = 50000437,50000466,50005823,50014578
TargetAcetylcholine receptor subunit epsilon(Homo sapiens (Human))
Guizhou Medical University
Curated by ChEMBL
Guizhou Medical University
Curated by ChEMBL
Affinity DataIC50: 2.30nMAssay Description:Inhibition of human AChE by Ellman's methodMore data for this Ligand-Target Pair
TargetAcetylcholine receptor subunit epsilon(Homo sapiens (Human))
Guizhou Medical University
Curated by ChEMBL
Guizhou Medical University
Curated by ChEMBL
Affinity DataIC50: 6nMAssay Description:Inhibition of AChE (unknown origin) after 2 minsMore data for this Ligand-Target Pair
TargetAcetylcholine receptor subunit epsilon(Homo sapiens (Human))
Guizhou Medical University
Curated by ChEMBL
Guizhou Medical University
Curated by ChEMBL
Affinity DataIC50: 12nMAssay Description:Inhibition of human AChE by Ellman's methodMore data for this Ligand-Target Pair
TargetAcetylcholine receptor subunit epsilon(Homo sapiens (Human))
Guizhou Medical University
Curated by ChEMBL
Guizhou Medical University
Curated by ChEMBL
Affinity DataIC50: 27nMAssay Description:Inhibition of AChE (unknown origin) after 2 minsMore data for this Ligand-Target Pair
TargetAcetylcholine receptor subunit epsilon(Homo sapiens (Human))
Guizhou Medical University
Curated by ChEMBL
Guizhou Medical University
Curated by ChEMBL
Affinity DataIC50: 32nMAssay Description:Inhibition of human AChE by Ellman's methodMore data for this Ligand-Target Pair
TargetAcetylcholine receptor subunit epsilon(Homo sapiens (Human))
Guizhou Medical University
Curated by ChEMBL
Guizhou Medical University
Curated by ChEMBL
Affinity DataIC50: 32nMAssay Description:Inhibition of human AChE by Ellman's methodMore data for this Ligand-Target Pair
TargetAcetylcholine receptor subunit epsilon(Homo sapiens (Human))
Guizhou Medical University
Curated by ChEMBL
Guizhou Medical University
Curated by ChEMBL
Affinity DataIC50: 36nMAssay Description:Inhibition of human AChE by Ellman's methodMore data for this Ligand-Target Pair
TargetAcetylcholine receptor subunit epsilon(Homo sapiens (Human))
Guizhou Medical University
Curated by ChEMBL
Guizhou Medical University
Curated by ChEMBL
Affinity DataIC50: 44nMAssay Description:Inhibition of human AChE by Ellman's methodMore data for this Ligand-Target Pair
TargetAcetylcholine receptor subunit epsilon(Homo sapiens (Human))
Guizhou Medical University
Curated by ChEMBL
Guizhou Medical University
Curated by ChEMBL
Affinity DataIC50: 44nMAssay Description:Inhibition of acetylcholinesteraseMore data for this Ligand-Target Pair
TargetAcetylcholine receptor subunit epsilon(Homo sapiens (Human))
Guizhou Medical University
Curated by ChEMBL
Guizhou Medical University
Curated by ChEMBL
Affinity DataIC50: 47nMAssay Description:Inhibition of AChE (unknown origin) by Ellman's methodMore data for this Ligand-Target Pair
TargetAcetylcholine receptor subunit epsilon(Homo sapiens (Human))
Guizhou Medical University
Curated by ChEMBL
Guizhou Medical University
Curated by ChEMBL
Affinity DataIC50: 50nMAssay Description:Inhibition of nAChR epsilon (unknown origin)More data for this Ligand-Target Pair
TargetAcetylcholine receptor subunit epsilon(Homo sapiens (Human))
Guizhou Medical University
Curated by ChEMBL
Guizhou Medical University
Curated by ChEMBL
Affinity DataIC50: 57nMAssay Description:Inhibition of AChE (unknown origin) by Ellman's methodMore data for this Ligand-Target Pair
TargetAcetylcholine receptor subunit epsilon(Homo sapiens (Human))
Guizhou Medical University
Curated by ChEMBL
Guizhou Medical University
Curated by ChEMBL
Affinity DataIC50: 58nMAssay Description:Inhibition of AChE (unknown origin) by Ellman's methodMore data for this Ligand-Target Pair
TargetAcetylcholine receptor subunit epsilon(Homo sapiens (Human))
Guizhou Medical University
Curated by ChEMBL
Guizhou Medical University
Curated by ChEMBL
Affinity DataIC50: 58nMAssay Description:Inhibition of human AChE by Ellman's methodMore data for this Ligand-Target Pair
TargetAcetylcholine receptor subunit epsilon(Homo sapiens (Human))
Guizhou Medical University
Curated by ChEMBL
Guizhou Medical University
Curated by ChEMBL
Affinity DataIC50: 62nMAssay Description:Inhibition of AChE (unknown origin) by Ellman's methodMore data for this Ligand-Target Pair
TargetAcetylcholine receptor subunit epsilon(Homo sapiens (Human))
Guizhou Medical University
Curated by ChEMBL
Guizhou Medical University
Curated by ChEMBL
Affinity DataIC50: 71nMAssay Description:Inhibition of human AChE by Ellman's methodMore data for this Ligand-Target Pair
TargetAcetylcholine receptor subunit epsilon(Homo sapiens (Human))
Guizhou Medical University
Curated by ChEMBL
Guizhou Medical University
Curated by ChEMBL
Affinity DataIC50: 82nMAssay Description:Inhibition of AChE (unknown origin)More data for this Ligand-Target Pair
TargetAcetylcholine receptor subunit epsilon(Homo sapiens (Human))
Guizhou Medical University
Curated by ChEMBL
Guizhou Medical University
Curated by ChEMBL
Affinity DataIC50: 83nMAssay Description:Inhibition of human AChE by Ellman's methodMore data for this Ligand-Target Pair
TargetAcetylcholine receptor subunit epsilon(Homo sapiens (Human))
Guizhou Medical University
Curated by ChEMBL
Guizhou Medical University
Curated by ChEMBL
Affinity DataIC50: 87nMAssay Description:Inhibition of human AChE by Ellman's methodMore data for this Ligand-Target Pair
TargetAcetylcholine receptor subunit epsilon(Homo sapiens (Human))
Guizhou Medical University
Curated by ChEMBL
Guizhou Medical University
Curated by ChEMBL
Affinity DataIC50: 88nMAssay Description:Inhibition of AChE (unknown origin) by Ellman's methodMore data for this Ligand-Target Pair
TargetAcetylcholine receptor subunit epsilon(Homo sapiens (Human))
Guizhou Medical University
Curated by ChEMBL
Guizhou Medical University
Curated by ChEMBL
Affinity DataIC50: 91nMAssay Description:Inhibition of human AChE by Ellman's methodMore data for this Ligand-Target Pair
TargetAcetylcholine receptor subunit epsilon(Homo sapiens (Human))
Guizhou Medical University
Curated by ChEMBL
Guizhou Medical University
Curated by ChEMBL
Affinity DataIC50: 97nMAssay Description:Inhibition of AChE (unknown origin) by Ellman's methodMore data for this Ligand-Target Pair
TargetAcetylcholine receptor subunit epsilon(Homo sapiens (Human))
Guizhou Medical University
Curated by ChEMBL
Guizhou Medical University
Curated by ChEMBL
Affinity DataIC50: 125nMAssay Description:Inhibition of acetylcholinesteraseMore data for this Ligand-Target Pair
TargetAcetylcholine receptor subunit alpha/beta/delta/epsilon(Homo sapiens)
Veterans Affairs Medical Center
Curated by ChEMBL
Veterans Affairs Medical Center
Curated by ChEMBL
Affinity DataIC50: 131nMAssay Description:Inhibition of human alpha1beta1deltaepsilon nAChR expressed in Xenopus laevis oocytes assessed as inhibition of acetylcholine-induced current respons...More data for this Ligand-Target Pair
TargetAcetylcholine receptor subunit epsilon(Homo sapiens (Human))
Guizhou Medical University
Curated by ChEMBL
Guizhou Medical University
Curated by ChEMBL
Affinity DataIC50: 407nMAssay Description:Inhibition of human AChE by Ellman's methodMore data for this Ligand-Target Pair
TargetAcetylcholine receptor subunit epsilon(Homo sapiens (Human))
Guizhou Medical University
Curated by ChEMBL
Guizhou Medical University
Curated by ChEMBL
Affinity DataIC50: 676nMAssay Description:Inhibition of human AChE by Ellman's methodMore data for this Ligand-Target Pair
TargetAcetylcholine receptor subunit epsilon(Rattus norvegicus)
Zhejiang Academy Of Medical Sciences
Curated by ChEMBL
Zhejiang Academy Of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of rat brain cortex AChE using acetylthiocholine iodide as substrate incubated for 15 mins by spectrophotometryMore data for this Ligand-Target Pair
TargetAcetylcholine receptor subunit epsilon(Homo sapiens (Human))
Guizhou Medical University
Curated by ChEMBL
Guizhou Medical University
Curated by ChEMBL
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibition of human AChE using acetylthiocholine iodide as substrate after 10 secs measured at 30 s intervals for two minutes by Ellman's methodMore data for this Ligand-Target Pair
TargetAcetylcholine receptor subunit epsilon(Homo sapiens (Human))
Guizhou Medical University
Curated by ChEMBL
Guizhou Medical University
Curated by ChEMBL
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibition of AChE (unknown origin)More data for this Ligand-Target Pair
TargetAcetylcholine receptor subunit epsilon(Homo sapiens (Human))
Guizhou Medical University
Curated by ChEMBL
Guizhou Medical University
Curated by ChEMBL
Affinity DataIC50: 2.66E+3nMAssay Description:Inhibition of AChE (unknown origin)More data for this Ligand-Target Pair
TargetAcetylcholine receptor subunit epsilon(Homo sapiens (Human))
Guizhou Medical University
Curated by ChEMBL
Guizhou Medical University
Curated by ChEMBL
Affinity DataIC50: 2.72E+3nMAssay Description:Inhibition of AChE (unknown origin)More data for this Ligand-Target Pair
TargetAcetylcholine receptor subunit epsilon(Homo sapiens (Human))
Guizhou Medical University
Curated by ChEMBL
Guizhou Medical University
Curated by ChEMBL
Affinity DataIC50: 3.06E+3nMAssay Description:Inhibition of AChE (unknown origin)More data for this Ligand-Target Pair
TargetAcetylcholine receptor subunit epsilon(Homo sapiens (Human))
Guizhou Medical University
Curated by ChEMBL
Guizhou Medical University
Curated by ChEMBL
Affinity DataIC50: 6.37E+3nMAssay Description:Inhibition of AChE (unknown origin)More data for this Ligand-Target Pair
TargetAcetylcholine receptor subunit epsilon(Rattus norvegicus)
Zhejiang Academy Of Medical Sciences
Curated by ChEMBL
Zhejiang Academy Of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 7.94E+3nMAssay Description:Inhibition of acetylcholinesterase in rat brain homogenate after 15 mins by Ellman assayMore data for this Ligand-Target Pair
TargetAcetylcholine receptor subunit epsilon(Homo sapiens (Human))
Guizhou Medical University
Curated by ChEMBL
Guizhou Medical University
Curated by ChEMBL
Affinity DataIC50: 8.00E+3nMAssay Description:Inhibition of AChE (unknown origin)More data for this Ligand-Target Pair
TargetAcetylcholine receptor subunit epsilon(Rattus norvegicus)
Zhejiang Academy Of Medical Sciences
Curated by ChEMBL
Zhejiang Academy Of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 8.30E+3nMAssay Description:Inhibition of rat brain cortex AChE using acetylthiocholine iodide as substrate incubated for 15 mins by spectrophotometryMore data for this Ligand-Target Pair
TargetAcetylcholine receptor subunit epsilon(Rattus norvegicus)
Zhejiang Academy Of Medical Sciences
Curated by ChEMBL
Zhejiang Academy Of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 8.80E+3nMAssay Description:Inhibition of rat brain cortex AChE using acetylthiocholine iodide as substrate incubated for 15 mins by spectrophotometryMore data for this Ligand-Target Pair
TargetAcetylcholine receptor subunit epsilon(Rattus norvegicus)
Zhejiang Academy Of Medical Sciences
Curated by ChEMBL
Zhejiang Academy Of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 9.00E+3nMAssay Description:Inhibition of rat brain cortex AChE using acetylthiocholine iodide as substrate incubated for 15 mins by spectrophotometryMore data for this Ligand-Target Pair
TargetAcetylcholine receptor subunit epsilon(Rattus norvegicus)
Zhejiang Academy Of Medical Sciences
Curated by ChEMBL
Zhejiang Academy Of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of acetylcholinesterase in rat brain homogenate after 15 mins by Ellman assayMore data for this Ligand-Target Pair
TargetAcetylcholine receptor subunit alpha/beta/delta/epsilon(MOUSE)
Hainan University
Curated by ChEMBL
Hainan University
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of dopamine uptake in rat synaptosomal fractionMore data for this Ligand-Target Pair
TargetAcetylcholine receptor subunit alpha/beta/delta/epsilon(MOUSE)
Hainan University
Curated by ChEMBL
Hainan University
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of mouse alpha1beta1deltaepsilon nAChR expressed in Xenopus laevis oocytes assessed as inhibition of ACh-induced current after 2 to 4 days...More data for this Ligand-Target Pair
TargetAcetylcholine receptor subunit alpha/beta/delta/epsilon(Homo sapiens)
Veterans Affairs Medical Center
Curated by ChEMBL
Veterans Affairs Medical Center
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human alpha1beta1deltaepsilon nAChR expressed in Xenopus laevis oocytes assessed as inhibition of acetylcholine-induced current respons...More data for this Ligand-Target Pair
TargetAcetylcholine receptor subunit epsilon(Rattus norvegicus)
Zhejiang Academy Of Medical Sciences
Curated by ChEMBL
Zhejiang Academy Of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 1.02E+4nMAssay Description:Inhibition of acetylcholinesterase in rat brain homogenate after 15 mins by Ellman assayMore data for this Ligand-Target Pair
TargetAcetylcholine receptor subunit epsilon(Homo sapiens (Human))
Guizhou Medical University
Curated by ChEMBL
Guizhou Medical University
Curated by ChEMBL
Affinity DataIC50: 1.23E+4nMAssay Description:Inhibition of AChE (unknown origin)More data for this Ligand-Target Pair
TargetAcetylcholine receptor subunit epsilon(Rattus norvegicus)
Zhejiang Academy Of Medical Sciences
Curated by ChEMBL
Zhejiang Academy Of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 1.36E+4nMAssay Description:Inhibition of rat brain cortex AChE using acetylthiocholine iodide as substrate incubated for 15 mins by spectrophotometryMore data for this Ligand-Target Pair
TargetAcetylcholine receptor subunit epsilon(Rattus norvegicus)
Zhejiang Academy Of Medical Sciences
Curated by ChEMBL
Zhejiang Academy Of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 1.63E+4nMAssay Description:Inhibition of rat brain cortex AChE using acetylthiocholine iodide as substrate incubated for 15 mins by spectrophotometryMore data for this Ligand-Target Pair
TargetAcetylcholine receptor subunit epsilon(Rattus norvegicus)
Zhejiang Academy Of Medical Sciences
Curated by ChEMBL
Zhejiang Academy Of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 1.81E+4nMAssay Description:Inhibition of rat brain cortex AChE using acetylthiocholine iodide as substrate incubated for 15 mins by spectrophotometryMore data for this Ligand-Target Pair
TargetAcetylcholine receptor subunit epsilon(Rattus norvegicus)
Zhejiang Academy Of Medical Sciences
Curated by ChEMBL
Zhejiang Academy Of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 1.95E+4nMAssay Description:Inhibition of acetylcholinesterase in rat brain homogenate after 15 mins by Ellman assayMore data for this Ligand-Target Pair
TargetAcetylcholine receptor subunit epsilon(Rattus norvegicus)
Zhejiang Academy Of Medical Sciences
Curated by ChEMBL
Zhejiang Academy Of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 2.06E+4nMAssay Description:Inhibition of rat brain cortex AChE using acetylthiocholine iodide as substrate incubated for 15 mins by spectrophotometryMore data for this Ligand-Target Pair
TargetAcetylcholine receptor subunit epsilon(Rattus norvegicus)
Zhejiang Academy Of Medical Sciences
Curated by ChEMBL
Zhejiang Academy Of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 2.29E+4nMAssay Description:Inhibition of acetylcholinesterase in rat brain homogenate after 15 mins by Ellman assayMore data for this Ligand-Target Pair